性能参数
产品名称
BRCA1-IN-2
规格
100mg 250mg 500mg
货号
GOY-Y3554
含量
>98.00%
CAS
1622262-55-8
别名
N/A
化学名
分子式
C26H33N4O7P
分子量
分子量 544.54
溶解度
Soluble in DMSO
储存条件
Store at -20°C
General tips
用途
仅供科研
价格
电询
详细内容
BRCA1-IN-2 (compound 15) is a cell-permeable protein-protein interaction (PPI) inhibitor for BRCA1 with an IC50 of 0.31 μM and a Kd of 0.3 μM, which shows antitumor activities via the disruption of BRCA1 (BRCT)2/protein interactions[1]. IC50: 0.31 μM (BRCA1)[1]Kd: 0.3 μM (BRCA1)[1]
[1]. Na Z, et al. Protein-Protein Interaction Inhibitors of BRCA1 Discovered Using Small Molecule Microarrays. Methods Mol Biol. 2017;1518:139-156.
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传真号码:021-39596320 021-39921927
QQ: 3004918891 3004905818 3004901493 移动电话:18321818584 15026555973 地址:上海松江新砖公路1155号
产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!