apimod tetrahydrochloride
如果您对该产品感兴趣的话,可以
产品名称:
apimod tetrahydrochloride
产品型号:
GOY-Y3410
产品展商:
谷研
产品文档:
无相关文档
发布时间:2023-05-08
简单介绍
D-Ribose 5-phosphate disodium dihydrateH2O: 100 mg/mL (322.48 mM); DMSO: 1 mg/mL (3.22 mM)
apimod tetrahydrochloride
的详细介绍
性能参数
|
产品名称
|
apimod tetrahydrochloride
|
规格
|
5mg
|
货号
|
GOY-Y3410
|
含量
|
>97.00%
|
CAS
|
164301-51-3
|
别名
|
N/A
|
|
|
化学名
|
N/A
|
分子式
|
C34H56Cl4N18O2
|
分子量
|
分子量 890.74
|
溶解度
|
Soluble in DMSO
|
储存条件
|
-20°C, protect from light
|
General tips
|
|
用途
|
仅供科研
|
价格
|
电询
|
|
详细内容
|
Semapimod tetrahydrochloride (CNI-1493), an inhibitor of proinflammatory cytokine production, can inhibit TNF-α, IL-1β, and IL-6. Semapimod tetrahydrochloride inhibits TLR4 signaling (IC50≈0.3 μM). Semapimod tetrahydrochloride inhibits p38 MAPK and nitric oxide production in macrophages. Semapimod tetrahydrochloride has potential in a variety of inflammatory and autoimmune disorders[1][2][3].
[1]. Nishimatsu H, et al. Blockade of endogenous proinflammatory cytokines ameliorates endothelial dysfunction in obese Zucker rats. Hypertens Res. 2008;31(4):737‐743. [2]. Wehner S, Set al. Inhibition of p38 mitogen-activated protein kinase pathway as prophylaxis of postoperative ileus in mice. Gastroenterology. 2009;136(2):619‐629. [3]. Wang J, et al. Experimental Anti-Inflammatory Drug Semapimod Inhibits TLR Signaling by Targeting the TLR Chaperone gp96. J Immunol. 2016;196(12):5130‐5137.
|
公司正在销售的产品:
二氧化硅 14808-60-7 L-2 4-DIAMINOBUTYRIC ACID MONOHYDRO-CHLO 1482-98-0
4-甲基吡啶-3-硼酸 148546-82-1 四正辛基溴化铵 14866-33-2
噻菌灵 148-79-8 5-氯-2-甲基苯硼酸 148839-33-2
4-(甲磺?;┍脚鹚? 149104-88-1 4-乙?;脚鹚? 149104-90-5
2-羧基苯硼酸 149105-19-1 2-巯基苯并噻唑 149-30-4
异辛酸 149-5?
|
Naphazoline-d4 (hydrochloride)500 μg 1 mg 5 mg>99.00%Cas No. N/AC14H10D4N2·HCl
1-Stearoyl-d35-2-hydroxy-sn-glycero-3-PC5 mg>99.00%Cas No. 327178-92-7C26H19D35NO7P
Amodiaquine-d101mg>99.00%Cas No. 1189449-70-4C20H12ClD10N3O
Imiquimod100mg>99.00%Cas No. 99011-02-6C14H16N4
Metronidazole-d41 mg>99.00%Cas No. 1261392-47-5C6H5D4N3O3
NG,NG-dimethyl-L-Arginine-d6 (hydrochloride)1mg>99.00%Cas No. 1313730-20-9C8H12D6N4O2?2HCl
(+)-β-Citronellol250mg 500mg>99.00%Cas No. 1117-61-9C10H20O
|