性能参数 |
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产品名称 |
Mivebresib |
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规格 |
2mg 5mg 10mg 25mg 50mg |
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货号 |
GOY-Y2992 |
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含量 |
>98.00% |
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CAS |
1445993-26-9 |
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别名 |
N/A |
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化学名 |
N/A |
分子式 |
C22H19F2N3O4S |
分子量 |
分子量 459.47 |
溶解度 |
DMSO : 100 mg/mL (217.64 mM) |
储存条件 |
Store at -20°C |
General tips |
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用途 |
仅供科研 |
价格 |
电询 |
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详细内容 |
Mivebresib is a potent and orally available bromodomain and extraterminal domain (BET) bromodomain inhibitor. Mivebresib binds to BRD4 with a Ki of 1.5 nM. Mivebresib inhibit DHT-stimulated transcription of AR target genes without significant effect on AR protein expression. In addition to blocking the transcription activation downstream of AR, Mivebresib is also a potent inhibitor of MYC and the TMPRSS2-ETS fusion proteins[1]. |
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产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!