性能参数
产品名称
SDZ 224-015
规格
5 mg 10 mg 25 mg
货号
GOY-Y2823
含量
>98.00%
CAS
161511-45-1
别名
N/A
化学名
分子式
C30H35Cl2N3O9
分子量
分子量 652.52
溶解度
储存条件
Store at -20°C
General tips
用途
仅供科研
价格
电询
详细内容
SDZ 224-015 is an orally active inhibitor of the interleukin-1 beta (IL-1β) converting enzyme and caspase-1. SDZ 224-015 possesses anti-COVID-19 activity, targeting Mpro (IC50 of 30 nM)[1][2].
SDZ 224-015 (0.3-300 μg/kg) potently reduces carrageenin-induced paw oedema[2].SDZ 224-015 (0.2-5 mg/kg, p.o.) displays analgesic activity in the Randall-Selitto yeast-inflamed paw pressure test, significant at a dose of 1 mg/kg[2].
[1]. Martin A Redhead, et al. Bispecific repurposed medicines targeting the viral and immunological arms of COVID-19. Sci Rep. 2021 Jun 24;11(1):13208.
[2]. P R Elford, et al. Reduction of inflammation and pyrexia in the rat by oral administration of SDZ 224-015, an inhibitor of the interleukin-1 beta converting enzyme. Br J Pharmacol. 1995 Jun;115(4):601-6.
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产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!