性能参数 |
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产品名称 |
RSM-932A |
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规格 |
1mg 5mg 10mg |
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货号 |
GOY-Y2814 |
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含量 |
>98.00% |
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CAS |
850807-63-5 |
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别名 |
N/A |
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化学名 |
1,1'-[[[1,1'-biphenyl]-4,4'-diyl]bis(methylene)]bis[4-[(4-chlorophenyl)methylamino]-quinolinium, dibromide |
分子式 |
C46H38Cl2N4.2Br |
分子量 |
分子量 877.5 |
溶解度 |
3mg/mL in DMSO |
储存条件 |
Store at -20°C |
General tips |
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用途 |
仅供科研 |
价格 |
电询 |
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详细内容 |
RSM-932A is a selective inhibitor of choline kinase α (CHOKα; IC50s = 1 and >50 μM for CHOKα and β, respectively). It induces apoptosis via CHOP signaling and endoplasmic reticulum (ER) stress in MDA-MB-231, MCF-7, SW620, and H460 cancer cells, but it only induces cell cycle arrest and not apoptosis in NCM460 and MCF-10A normal epithelial cells.[2] RSM-932A inhibits the growth of HT-29 colon cancer cells in vitro (IC50 = 1.15 μM) and in vivo in a mouse xenograft model (ED50 = 7.5 mg/kg). [1] |
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产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!