性能参数 |
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产品名称 |
OD 36 hydrochloride |
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规格 |
10 mg |
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货号 |
GOY-Y2572 |
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含量 |
>98.00% |
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CAS |
1638644-62-8 |
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别名 |
N/A |
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化学名 |
N/A |
分子式 |
C16H15ClN4O2.HCl |
分子量 |
分子量 367.23 |
溶解度 |
Soluble in DMSO |
储存条件 |
Desiccate at RT |
General tips |
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用途 |
仅供科研 |
价格 |
电询 |
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详细内容 |
Potent receptor-interacting protein kinase 2 (RIPK2) inhibitor (IC50 = 5.3 nM). Displays similar % inhibition against ALK-2 and SIK2 at 100 nM. Downregulates expression of a panel of RIPK2-dependent genes. Inhibits recruitment of inflammatory cells in a mouse MDP-induced peritonitis model. Tigno-Aranjuez et al (2014) In vivo inhibition of RIPK2 kinase alleviates inflammatory disease. J.Biol.Chem. 289 29651 PMID:25213858 |Sánchez-Duffhues et al (2019) Development of macrocycle kinase inhibitors for ALK2 using Fibrodysplasia ossificans progressiva-derived endothelial cells. JBMRPlus 3 e10230 PMID:31768489 |
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