性能参数
产品名称
Diazepinomicin
规格
100mg 250mg
货号
GOY-Y2035
含量
>98.00%
CAS
733035-26-2
别名
N/A
化学名
分子式
C28H34N2O4
分子量
分子 462.58
溶解度
Soluble in DMSO
储存条件
Store at -20°C, protect from light, stored under nitrogen
General tips
用途
仅供科研
价格
电询
详细内容
Diazepinomicin (TLN-4601) is a secondary metabolite produced by Micromonospora sp. Diazepinomicin (TLN-4601) inhibits the EGF-induced Ras-ERK MAPK signaling pathway and induces apoptosis. An anti-tumor agent for K-Ras mutant models[1]. Diazepinomicin (TLN-4601) inhibits the EGF-induced Ras-ERK MAPK signaling pathway post Ras prenylation and prior to MEK activation[1].
[1]. Campbell PM, et al. TLN-4601 suppresses growth and induces apoptosis of pancreatic carcinoma cells through inhibition of Ras-ERK MAPK signaling. J Mol Signal. 2010 Nov 2;5:18.
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Purity: >97.00%
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产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!